Inventor
Jacob Szmuszkovicz
Inventor
Kalamazoo, MI, US
Overview
Patents· 40 as inventor
Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.
C07Dprimary
C07DHeterocyclic compounds47%
C07CAcyclic or carbocyclic compounds25%
A61PSpecific therapeutic activity of chemical compounds or medicinal preparations14%
A61KPreparations for medical, dental or toiletry purposes8%
C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium6%
PatentTitleYear
6,436,954'Benzoquinolizidine and benzoindolizidine derivatives and therapeutic uses thereof'20024,978,753'7-phenylpyrimido[1,2-alpha][1,4]benzodiazepin-3(5H)-ones'19904,801,604'Cis-N-(2-aminocycloaliphatic)benzamide anti-convulsants'19894,652,559'2-(Phenylmethylene)cycloalkyl-azetidines'19874,598,088'2-pyrrolyl-cycloalkyl-amide analgesics'19864,590,187'Phospholipase A.sub.2 inhibition using 4,1-benzoxazepine-2-(3H)-ones'19864,540,690'2-(Phenylmethylene)cycloalkylamines and -azetidines'19854,466,977'N-[2-Amino(oxy- or thia- group-substituted-cycloaliphatic)]benzeneacetamides and -benzamide analgesics'19844,460,600'Adjacently substituted ketal derivatives of cycloalkane-amide analgesics'19844,360,531'Substituted cycloalkanes'19824,359,476'Adjacently substituted cycloalkane-amide analgesics'1982RE030837'N-(2-Aminocycloheptyl)alkanoylanilides'19814,286,106'N-[.omega.-(Dimethylamino)alkyl]-3\',4\'-dichloropropionanilides'19814,217,362'Anilide derivatives as antidepressants'19804,215,114'Analgesic N-[2-(furyl-methylamino and 2-thienylmethylamino)cycloaliphatic]b e'19804,212,878'Phenylacetamide derivative analgesics'19804,212,888'Anilide derivatives as antidepressants'19804,204,003'N-(2-Aminocyclopentyl)-N-alkanoylanilides as CNS anti-depressants'19804,199,589'N-(2-Aminocycloheptyl)acylanilides and methods to treat depression'19804,197,308'Analgesic N-(2-heterocyclic-amino cycloaliphatic) benzamides'19804,192,885'Analgesic N-{2-[N\'-(2-furylmethyl and 2-thienyl-methyl)-N\'-alkylamino]cycloaliphatic}cyanobenzamides'19804,186,208'Anti-depressant N-(3,4-dichlorophenyl)-N-dimethylaminoalkylene amides'19804,180,522'N-(2-Dimethylaminoalkyl)-3\',4\'-dichloroanilides'19794,179,501'Analgesic N-(2-aminocycloaliphatic)azidobenzamides'19794,172,898'N-(2-aminocycloheptyl)acylanilides'19794,169,156'N-(2-aminocycloheptyl)alkanoylanilides'19794,159,339'N-(2-Aminocycloheptyl) alkanoylanilides'19794,159,340'N-(2-Aminocyclopentyl)-N-acylanilides as CNS anti-depressants'19794,157,398'N-(2-Aminocyclopentyl)acylanilides and treating depression'19794,156,733'N-(2-Aminocyclopentyl) alkanoylanilides'19794,156,015'N-(2-Aminocyclopentyl)acylanilides and treating depression'19794,156,014'N-(2-aminocycloheptyl)alkanoylanilides and in the treatment of depression'19794,153,717'Analgesic N-(2-(furylmethylamino and 2 -thienylmethylamino)cyclo aliphatic)benzamides'19794,152,459'Analgesic N-2-(aminocycloaliphatic)-hydroxy, alkoxy and (allylic)alkenyloxy-benzamides'19794,148,914'Analgesic N-(2-aminocyclo aliphatic)cyanobenzamides'19794,145,435'2-Aminocycloaliphatic amide compounds'19794,128,663'Anilide derivatives as antidepressants'19784,098,904'Analgesic N-(2-aminocycloaliphatic)benzamides'19783,966,736'2,9-Dihydro-3H-pyrido[3,2-c]-s-triazolo[4,3-a][1,5]-benzodiazepin-3-ones'19763,933,816'3-(Substituted aminomethyl)-7-substituted-3,5-dihydro-as-triazino[4,3-a][1,5]benzodiaze pines'1976Career & activity timeline
Assembled from patent assignee/location history and declaration credentials.
1976–1990Patents assigned to UPJOHN CO (37)· patent assignee history
1976–2002Based in Kalamazoo, MI, US· patent location history
1980Patents assigned to SZMUSZKOVICZ JACOB (1)· patent assignee history
2002Patents assigned to AMERICAN BIOGENETIC SCIENCES (1)· patent assignee history
2002Patents assigned to UNIV DUBLIN (1)· patent assignee history
Inventor activity
Assignee and location history derived from the patent record.
Assignees
| Assignee | Patents | Span |
|---|---|---|
| UPJOHN CO | 37 | 1976–1990 |
| AMERICAN BIOGENETIC SCIENCES | 1 | 2002 |
| SZMUSZKOVICZ JACOBself | 1 | 1980 |
| UNIV DUBLIN | 1 | 2002 |
Locations
| Location | Patents | Span |
|---|---|---|
| Kalamazoo, MI, US | 40 | 1976–2002 |