Inventor
Dirk Kosemund
Inventor
Berlin, DE
Overview
Patents· 41 as inventor
Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.
A61Pprimary
A61PSpecific therapeutic activity of chemical compounds or medicinal preparations32%
C07DHeterocyclic compounds29%
A61KPreparations for medical, dental or toiletry purposes27%
C07JSteroids5%
C07CAcyclic or carbocyclic compounds3%
C07BGeneral methods of organic chemistry2%
C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium1%
C07KPeptides1%
Y02ATechnologies for adaptation to climate change1%
PatentTitleYear
10,428,083Heterocyclylmethyl-thienouracile as antagonists of the adenosine-A2B-receptor20199,962,3894-aryl-N-phenyl-1,3,5-triazin-2-amines containing a sulfoximine group20189,902,716'Fluorinated benzofuranyl-pyrimidine derivatives containing a sulfone group'20189,884,849'Fluorinated benzofuranyl-pyrimidine derivatives containing a sulfoximine group'20189,877,954'5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfoximine group'20189,856,242'5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfone group'20189,770,445'Sulfoximine substituted 5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives and their use as CDK9 kinase inhibitors'20179,708,293'N-(pyridin-2-yl)pyrimidin-4-amine derivatives containing a sulfone group'20179,676,766'Triazolopyridines'20179,669,034'4-aryl-N-phenyl-1,3,5-triazin-2-amines containing a sulfoximine group'20179,670,161'5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfone group'20179,670,202'Substituted triazolopyridines'20179,663,510'Substituted triazolopyridines and their use as TTK inhibitors'20179,650,361'N-(pyridin-2-yl)pyrimidin-4-amine derivatives containing a sulfoximine group'20179,650,340'5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfoximine group'20179,586,958'Prodrug derivatives of substituted triazolopyridines'20179,555,022'Substituted triazolopyridines'20179,540,392'Thienopyrimidines'20179,499,492'4-(ortho)-fluorophenyl-5-fluoropyrimidin-2-yl amines containing a sulfoximine group'20169,468,642'Imidazopyrazines'20169,388,140'Substituted benzimidazoles'20169,296,757'Substituted benzothienopyrimidines'20169,284,317'Substituted imidazo[1,2-a]pyrazines as MPS-1 inhibitors'20169,255,100'Substituted imidazopyridazines'20169,212,184'6-thio-substituted imidazo[1,2-a]pyrazines as Mps-1 inhibitors'20159,199,999'Substituted imidazopyrazines'20159,133,171'Disubstituted 5-fluoro pyrimidine derivatives containing a sulfoximine group'20159,108,926'Disubstituted 5-fluoro-pyrimidines'20158,916,557'Substituted 4-Aryl-N-phenyl-1,3,5-triazin-2-amines'20148,841,311'Sulphone-substituted quinazoline derivatives as immuno-modulators, their preparation and use as medicaments'20148,551,980'Substituted triazolopyridines'20138,492,570'2-substituted estra-1,3,5(10)-triene-3-yl sulfamate with an anti-tumor action'20137,511,059'Thiazolidinones, their production and use as pharmaceutical agents'20097,504,410'Chk-, Pdk- and Akt-inhibitory pyrimidines, their production and use as pharmaceutical agents'20097,449,459'Inhibitors of soluble adenylate cyclase'20087,427,610'2-substituted estra-1,3,5(10)-triene-3-yl sulfamate with an anti-tumour action'20087,414,043'9-α-substituted estratrienes as selectively active estrogens'20087,109,360'16-hydroxyestratrienes as selectively active estrogens'20066,794,409'Use of ER-selective ligands for regulating fertility and compounds useful therefor'20046,670,347'19-nor-17-pregna-1,3,5(10)-trien-17-ols with a 21,16-lactone ring'20036,583,130'C13-substituted estra-1,3,5,(10)-trien-3-yl sulfamates, methods of preparing same, and pharmaceutical compositions containing these compounds'2003Career & activity timeline
Assembled from patent assignee/location history and declaration credentials.
2003–2013Based in Erfurt, DE· patent location history
2013–2018Patents assigned to BAYER IP GMBH (16)· patent assignee history
2013–2017Patents assigned to KOSEMUND DIRK (15)· patent assignee history
2013–2017Patents assigned to SIEMEISTER GERHARD (14)· patent assignee history
2013–2017Patents assigned to LIENAU PHILIP (12)· patent assignee history
2013–2019Based in Berlin, DE· patent location history
2016–2019Patents assigned to Bayer Pharma AG (15)· patent assignee history
Inventor activity
Assignee and location history derived from the patent record.
Assignees
| Assignee | Patents | Span |
|---|---|---|
| BAYER IP GMBH | 16 | 2013–2018 |
| Bayer Pharma AG | 15 | 2016–2019 |
| KOSEMUND DIRKself | 15 | 2013–2017 |
| SIEMEISTER GERHARD | 14 | 2013–2017 |
| LIENAU PHILIP | 12 | 2013–2017 |
Locations
| Location | Patents | Span |
|---|---|---|
| Berlin, DE | 31 | 2013–2019 |
| Erfurt, DE | 10 | 2003–2013 |