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Inventor

Nicholas D. P. Cosford

Inventor
La Jolla, CA, US

Overview

39→
Patents
1996–2021
Patent span
Chemistry
Primary field (CPC C)

Patents· 39 as inventor

Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.

C07Dprimary
C07DHeterocyclic compounds32%
A61PSpecific therapeutic activity of chemical compounds or medicinal preparations24%
A61KPreparations for medical, dental or toiletry purposes14%
C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium10%
C07KPeptides6%
Y02ATechnologies for adaptation to climate change4%
C12QMeasuring or testing processes involving enzymes, nucleic acids or microorganisms3%
C12YEnzymes3%
G01NInvestigating or analysing materials by determining their chemical or physical properties3%
C07CAcyclic or carbocyclic compounds2%
PatentTitleYear
11,111,270Inhibitor of apoptosis protein (IAP) antagonists202110,864,217Use of inhibitor of apoptosis protein (IAP) antagonists in HIV therapy202010,774,092ULK1 inhibitors and methods using same202010,689,397ULK1 inhibitors and methods using same202010,597,367Metabotropic glutamate receptor negative allosteric modulators (NAMs) and uses thereof202010,544,188Inhibitor of apoptosis protein (IAP) antagonists202010,377,695Metabotropic glutamate receptor positive allosteric modulators (PAMS) and uses thereof201910,300,074Use of inhibitor of apoptosis protein (IAP) antagonists in HIV therapy201910,266,549ULK1 inhibitors and methods using same201910,099,993Metabotropic glutamate receptor positive allosteric modulators (PAMS) and uses thereof201810,071,976Small molecule fatty acid synthase inhibitors201810,047,119Inhibitor of apoptosis protein (IAP) antagonists20189,969,726Metabotropic glutamate receptor negative allosteric modulators (NAMS) and uses thereof20189,546,174'Inhibitor of apoptosis protein (IAP) antagonists'20177,592,337'Di-aryl substituted tetrazole modulators of metabotropic glutamate receptor-5'20097,589,068'Inhibitors of Akt activity'20097,569,592'Heteroaryl substituted pyrazole modulators of metabotropic glutamate receptor-5'20097,544,677'Inhibitors of Akt activity'20097,462,619'Pyridazine, pyrimidine and pyrazine ethyne compounds'20087,393,959'Di-aryl substituted pyrrole modulators of metabotropic glutamate receptor-5'20087,371,767'Heteroaryl substituted pyrrole modulators of metabotropic glutamate receptor-5'20087,365,074'Pyridazine, pyrimidine and pyrazine ethyne compounds'20087,268,151'Di-aryl substituted triazole modulators of metabotropic glutamate receptor-5'20077,253,190'Heteroaryl substituted tetrazole modulators of metabotrophic glutamate receptor-5'20077,105,548'Heteroaryl substituted triazole modulators of metabotropic glutamate receptor-5'20066,956,049'Methods of modulating processes mediated by excitatory amino acid receptors'20056,774,138'Thiazolyl(pyridyl)ethyne compounds'20046,656,957'Pyridine derivatives'20036,632,823'Substituted pyridine compounds useful as modulators of acetylcholine receptors'20036,194,581'Substituted pyridines useful as modulators of acetylcholine receptors'20015,852,041'Substituted pyridines useful as modulators of acethylcholine receptors'19985,736,560'Substituted pyridines useful as modulators of acetylcholine receptors'19985,723,477'Modulators of acetylcholine receptors'19985,705,512'Modulators of acetylcholine receptors'19985,703,100'Modulators of acetylcholine receptors'19975,686,473'Substituted pyridines useful as modulators of acetylcholine receptors'19975,677,459'Methods for the preparation of modulators of acetylcholine receptors'19975,594,011'Modulators of acetylcholine receptors'19975,585,388'Substituted pyridines useful as modulators of acetylcholine receptors'1996

Career & activity timeline

Assembled from patent assignee/location history and declaration credentials.

1996–2003Patents assigned to SIBIA NEUROSCIENCES INC (10)· patent assignee history
1996–2021Based in La Jolla, CA, US· patent location history
1997–2009Based in San Diego, CA, US· patent location history
2001–2009Patents assigned to MERCK & CO INC (15)· patent assignee history
2018–2021Patents assigned to SANFORD BURNHAM PREBYS MEDICAL DISCOVERY INST (10)· patent assignee history
2018–2019Patents assigned to SANFORD BURNHAM MED RES INST (4)· patent assignee history
2019–2020Patents assigned to SALK INST FOR BIOLOGICAL STUDI (5)· patent assignee history

Inventor activity

Assignee and location history derived from the patent record.

Assignees
AssigneePatentsSpan
MERCK & CO INC152001–2009
SANFORD BURNHAM PREBYS MEDICAL DISCOVERY INST102018–2021
SIBIA NEUROSCIENCES INC101996–2003
SALK INST FOR BIOLOGICAL STUDI52019–2020
SANFORD BURNHAM MED RES INST42018–2019
Locations
LocationPatentsSpan
La Jolla, California, US201996–2021
San Diego, California, US191997–2009