Inventor
Jeffrey J. Hale
Inventor
Westfield, NJ, US
Overview
Patents· 42 as inventor
Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.
C07Dprimary
C07DHeterocyclic compounds42%
A61PSpecific therapeutic activity of chemical compounds or medicinal preparations33%
A61KPreparations for medical, dental or toiletry purposes8%
C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium8%
C07CAcyclic or carbocyclic compounds5%
B60RVehicles, vehicle fittings, or vehicle parts, not otherwise provided for4%
PatentTitleYear
9,365,539'Prolylcarboxypeptidase inhibitors'20168,921,555'Substituted-1,3,8-triazaspiro[4.5]decane-2,4-diones'20148,815,865'Substituted 4-hydroxypyrimidine-5-carboxamides'20148,492,398'Spiroazaindoles'20138,445,680'Tetrahydrothieno pyridines'20138,372,863'Tetrahydro-1H-pyrrolo fused pyridones'20138,372,857'Substituted 4-hydroxypyrimidine-5-carboxamides'20138,354,403'Pyrrolidine derived beta 3 adrenergic receptor agonists'20138,309,544'Spiroindalones'20128,278,304'Substituted 4-hydroxypyrimidine-5-carboxamides'20127,999,107'Substituted pyrano[2,3-B]pyridine derivatives as cannabinoid-1 receptor modulators'20117,906,652'Heterocycle-substituted 3-alkyl azetidine derivatives'20117,659,294'2-(aryl)azacyclylmethyl carboxylates, sulfonates, phosphonates, phosphinates and heterocycles as S1P receptor agonists'20107,605,171'(3,4-disubstituted)propanoic carboxylates as S1P (Edg) receptor agonists'20097,479,504'Edg receptor agonists'20097,351,725'N-(benzyl)aminoalkylcarboxylates, phosphinates, phosphonates and tetrazoles as Edg receptor agonists'20087,309,721'Aminoalkylphosphonates and related compounds as Edg receptor agonists'20077,220,734'1-(amino)indanes and (1,2-dihydro-3-amino)-benzofurans, benzothiophenes and indoles as Edg receptor agonists'20077,199,142'1-((5-aryl-1,2,4-oxadiazol-3-yl) benzyl)azetidine-3-carboxylates and 1-((5-aryl-1,2,4-oxadiazol-3-yl)benzyl) pyrrolidine-3-carboxylates as edg receptor agonists'20077,125,887'Pyrrolidine modulators of CCR5 chemokine receptor activity'20066,638,930'Morpholine and thiomorpholine tachykinin receptor antagonists'20036,498,161'Pyrrolidine modulators of chemokine receptor activity'20026,399,619'Pyrrolidine modulators of chemokine receptor activity'20026,265,434'Pyrrolidine modulators of chemokine receptor activity'20016,248,755'Pyrrolidine modulators of chemokine receptor activity'20016,235,735'Morpholine and thiomorpholine tachykinin receptor antagonists'20016,166,037'Pyrrolidine and piperidine modulators of chemokine receptor activity'20006,048,859'Morpholine and thiomorpholine tachykinin receptor antagonists'20005,922,706'Morpholine and thiomorpholine tachykinin receptor antagonists'19995,877,191'Phenyl spiroethercycloalkyl tachykinin receptor antagonists'19995,872,116'Morpholine and thiomorpholine tachykinin receptor antagonists'19995,869,496'Spiro-substituted azacycles as tachykinin receptor antagonists'19995,780,467'Morpholine compounds are prodrugs useful as tachykinin receptor antagonists'19985,750,549'Cycloalkyl tachykinin receptor antagonists'19985,747,485'Substituted azetidiones as anti-inflammatory and antidegenerative agents'19985,719,147'Morpholine and thiomorpholine tachykinin receptor antagonists'19985,716,942'Treatment of migraine with morpholine tachykinin receptor antagonists'19985,691,336'Morpholine compounds are prodrugs useful as tachykinin receptor antagonists'19975,637,699'Process for preparing morpholine tachykinin receptor antagonists'19975,591,737'Substituted azetidinones as anti-inflammatory and antidegenerative agents'19975,512,570'Treatment of emesis with morpholine tachykinin receptor antagonists'19965,391,819'Process of making chiral 2-aryl-1,4-butanediamine derivatives as useful neurokinin-A antagonists'1995Career & activity timeline
Assembled from patent assignee/location history and declaration credentials.
1995–2010Patents assigned to MERCK & CO INC (30)· patent assignee history
1995–2016Based in Westfield, NJ, US· patent location history
2011–2016Patents assigned to MERCK SHARP & DOHME (12)· patent assignee history
2012–2016Patents assigned to HALE JEFFREY J (10)· patent assignee history
2012–2014Patents assigned to DEBENHAM JOHN S (5)· patent assignee history
2012–2014Patents assigned to CLEMENTS MATTHEW J (4)· patent assignee history
Inventor activity
Assignee and location history derived from the patent record.
Assignees
| Assignee | Patents | Span |
|---|---|---|
| MERCK & CO INC | 30 | 1995–2010 |
| MERCK SHARP & DOHME | 12 | 2011–2016 |
| HALE JEFFREY Jself | 10 | 2012–2016 |
| DEBENHAM JOHN S | 5 | 2012–2014 |
| CLEMENTS MATTHEW J | 4 | 2012–2014 |
Locations
| Location | Patents | Span |
|---|---|---|
| Westfield, New Jersey, US | 42 | 1995–2016 |