Inventor

David T. Connor

Inventor

Ann Arbor, MI, US

Overview

1976–2007

Patent span

Chemistry

Primary field (CPC C)

Patents· 151 as inventor

Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.

C07Dprimary

C07DHeterocyclic compounds55%

A61PSpecific therapeutic activity of chemical compounds or medicinal preparations17%

C07CAcyclic or carbocyclic compounds11%

A61KPreparations for medical, dental or toiletry purposes10%

C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium2%

C07GCompounds of unknown constitution1%

C40BCombinatorial chemistry1%

Y02PClimate change mitigation technologies in the production or processing of goods1%

C07KPeptides0%

C12PFermentation or enzyme-using processes to synthesise a desired chemical compound or composition or to separate optical isomers from a racemic mixture0%

PatentTitleYear

7,214,712'Isophthalic acid derivatives as matrix metalloproteinase inhibitors'2007 7,067,538'MCP-1 receptor antagonists and methods of use thereof'2006 7,015,237'Pyridine matrix metalloproteinase inhibitors'2006 6,995,151'Isophthalic acid derivatives as matrix metalloproteinase inhibitors'2006 6,881,743'Pyridine matrix metalloproteinase inhibitors'2005 6,858,739'Indole and benzimidazole 15-lipoxygenase inhibitors'2005 6,548,499'Substituted quinoxaline derivatives as interleukin-8 receptor antagonists'2003 6,534,521'2-phenyl benzimidazole derivatives as MCP-1 antagonists'2003 6,528,528'Thiourea and benzamide compounds, compositions and methods of treating or preventing inflammatory diseases and atherosclerosis'2003 6,458,806'Aryl alkenamides derivatives as MCP-1 antagonists'2002 6,458,781'Substituted diarylalkyl amides as calcium channel antagonists'2002 6,423,689'Peptidyl calcium channel blockers'2002 6,348,487'2-phenyl benzimidazole derivatives as MCP-1 antagonists'2002 6,268,387'Thiourea and benzamide compounds, compositions and methods of treating or preventing inflammatory diseases and atherosclerosis'2001 6,211,209'Method of inhibiting connective tissue degradation'2001 6,184,235'2-phenyl benzimidazole derivatives as MCP-1 antagonists'2001 6,162,830'Benzenesulfonamide inhibitors of PDE-IV and their therapeutic use'2000 6,051,605'Method of treating psychosis and schizophrenia'2000 6,020,364'Compounds and method of treating psychosis and schizophrenia'2000 5,916,914'Compounds and method of treating psychosis and schizophrenia'1999 5,760,050'Antipsychotic method utilizing certain tetrahydrochromeno›3,4-c!pyridin-5-ones'1998 5,703,069'Method for inhibiting and controlling viral growth'1997 5,703,119'Benzylidene-lactone derivatives of fenamates and their thiocarbonyl analogs as inhibitors of proteoglycan degradation'1997 5,612,330'Methods for inhibiting and controlling viral growth'1997 5,571,825'Method of selectively inhibiting prostaglandin G/H synthase-2'1996 5,565,446'Benzothiophene, benzofuran and indole-thiazepinones, oxazepinones and diazepinones as inhibitors of cell adhesion and as inhibitors of HIV'1996 5,494,927'3,5-di-tertiarybutyl-4-hydroxyphenylmethylene derivatives of 2-substituted thiazolidinones, oxazolidinones, and imidazolidinones as antiinflammatory agents'1996 5,489,598'Cytoprotection utilizing aryltriazol-3-thiones'1996 5,489,586'Method for treating inflammatory disease in humans'1996 5,464,856'Arylmethylenyl derivatives of imidazolidinones useful as antiinflammatory agents'1995 5,464,855'Thiophene-2-carboxamidotetrazoles and pharmaceutical use thereof'1995 5,462,952'Fenamate 1,3,4-thiadiazoles and 1,3,4-oxadiazoles as antiinflammatory agents'1995 5,444,085'Methods of inhibiting HIV and inhibiting the activation of HIV'1995 5,434,188'1-ether and 1-thioether-naphthalene-2-carboxamides as inhibitors of cell adhesion and as inhibitors of the activation of HIV'1995 5,432,181'Substituted heteroaryl analogs of 4,6-di-tertiary-butyl-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents'1995 5,424,329'Indole-2-carboxamides as inhibitors of cell adhesion'1995 5,393,923'3,5-di-t-butyl-4-hydroxyphenylmethylhydroxylamines and their derivatives, pharmaceutical compositions, and methods of use therefor'1995 5,376,670'3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxyphenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents'1994 5,358,964'Benzylidene-lactone and their thiocarbonyl analogs as inhibitors of proteoglycan degradation'1994 5,356,898'Substituted 4,6-di-tertiary-butyl 5-hydroxy-pyrimidines'1994 5,356,926'3-alkyloxy-, aryloxy-, or arylalkyloxy-benzo [.beta.]thiophene-2-carboxamides as inhibitors of cell adhesion'1994 5,350,748'3-thio or amino substituted-benzo[b]thiophene-2-carboxamides and 3-oxygen, thio, or amino substituted-benzofuran-2-carboxamides as inhibitors of cell adhesion'1994 5,348,957'5-hydroxy-2-pyrimidinylmethylene derivatives useful as antiinflammatory agents'1994 5,340,815'2-substituted-4,6-di-tertiary-butyl-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents'1994 5,338,737'Biphenyl oxadiazoles and thiadiazoles as angiotensin II antagonists'1994 5,312,821'2-heterocyclic-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents'1994 5,306,822'Arylmethylenyl derivatives of oxazolidinone'1994 5,302,597'2-substituted-4,6-di-tertiarybutyl-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents'1994 5,290,800'3,5-di-tertiarybutyl-4-hydroxyphenylmethylene derivatives of 2-substituted thiazolidinones, oxazolidinones, and imidazolidinones as antiinflammatory agents'1994 5,288,896'3,5-di-t-butyl-4-hydroxylphenylmethylhydroxylamines and their derivatives, pharmaceutical compositions, and methods of use therefor'1994 5,284,949'2-substituted amino-4,6-di-tertiary-butyl-5-hydroxy-1,3-pyrimidines as antiinflammatory agents'1994 5,270,319'5-hydroxy-2-pyrimidinylmethylene derivatives useful as antiinflammatory agents'1993 5,256,680'3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxy-phenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents'1993 5,250,552'3-[thiazolidinone, oxazolidinone, imidazolidinone]-indoles as antiinflammatory agents'1993 5,248,682'2-substituted-4,6-di-tertiary-butyl-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents'1993 5,240,929'2-heterocyclic-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents'1993 5,234,937'3,5-di-tertiary-butyl-4-hydroxphenyl oxazolyl methanones and related compounds as antiinflammatory agents'1993 5,234,939'3,5-di-tertiary-butyl-4-hydroxyphenyl imidazolyl methanones and related compounds as antiinflammatory agents'1993 5,220,025'2-substituted amino-4, 6-di-tertiary-butyl-5-hydroxy-1, 3-pyrimidines as antiinflammatory agents'1993 5,215,986'5-hydroxy-2-pyrimidinylmethylene oxaza heterocycles'1993 5,212,189'Thiadiazole or oxadiazole analogs of fenamic acids containing substituted hydroxamate side chains as antiinflammatory agents'1993 5,210,204'Biphenyl oxadiazoles and thiadiazoles as angiothesin II antagonists'1993 5,208,253'3-alkyloxy-, aryloxy-, or arylalkyloxy-benzo(b) thiophene-2-carboxamides as inhibitors of cell adhesion'1993 5,208,251'Styryl pyrazoles, isoxazoles and analogs thereof having activity as 5-lipoxygenase inhibitors, pharmaceutical compositions and methods of use therefor'1993 5,208,250'Known and selected novel arylmethylenyl derivatives of thiazolidinones, imidazolidinones and oxazolidinones useful as antiallergy agents and anti-inflammatory agents'1993 5,196,431'2-substituted amino-4, 6-di-tertiary-buthyl-5-hydroxy-1, 3-pyrimidines as antiinflammatory agents'1993 5,187,175'2-carbonyl substituted-5-hydroxy-1, 3-pyrimidines as antiinflammatory agents'1993 5,177,259'Diarylalkanoids having activity as lipoxygenase inhibitors'1993 5,177,079'2-substituted-4,6-di-tertiarybutyl-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents'1993 5,155,110'Fenamic acid hydroxamate derivatives having cyclooxygenase and 5-lipoxygenase inhibition'1992 5,155,122'3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxy-phenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents'1992 5,143,927'3-(thiazolidone, oxazolidinone, imidazolidinone)-indoles as antiinflammatory agents'1992 5,143,929'2-substituted thiazolidinone, oxazolidinone, and imidazolidinone derivatives of fenamates as antiinflammatory agents'1992 5,143,928'3,5-di-tertiarybutyl-4-hydroxyphenylmethylene derivatives of 2-substituted thiazolidinones, oxazolidinones, and imidazolidinones as antiinflammatory agents'1992 5,142,095'Diarylalkanoids having activity as lipoxygenase inhibitors'1992 5,124,347'3-5-ditertiarybutylphenyl-4-hydroxymethylidene derivatives of 1,3-dihydro-2H-indole-2-ones as antiinflammatory agents'1992 5,114,958'1,2,4-oxadiazole and 1,2,4-thiadiazole derivatives of fenamates as antiinflammatory agents'1992 5,112,868'Hydroxamate derivatives of selected nonsteroidal antiinflammatory acyl residues having cyclooxygenase and 5-lipoxygenase inhibition'1992 5,112,846'N-hydroxyamide, N-hydroxythioamide, hydroxyurea, and N-hydroxythiourea derivatives of selected nsaids as antiinflammatory agents'1992 5,102,897'3,5-ditertiarybutyl-4-hydroxyphenyl, 1,3,4-thiadiazoles and oxadiazoles linked by carbon, oxygen, and sulfur residues'1992 5,086,064'3,5-di-tertiary-butyl-4-hydroxyphenyl thiazolyl, oxazolyl, and imidazolyl methanones and related compounds as antiinflammatory agents'1992 5,077,411'Dairylalkanoids having activity as lipoxygenase inhibitors'1991 5,075,330'N-hydroxyamide, N-hydroxythioamide, N-hydroxyurea, and N-hydroxythiourea derivatives of selected NSAIDS as antiinflammatory agents'1991 5,066,668'Triazole derivatives of fenamates as antiinflammatory agents'1991 4,981,865'N-hydroxyamide, N-hydroxythioamide, hydroxyurea, and N-hydroxythiourea derivatives of selected nsaids as antiinflammatory agents'1991 4,962,119'Triazole derivatives of fenamates as antiinflammatory agents'1990 4,959,503'Diarylalkanoids having activity as lipoxygenase inhibitors'1990 4,943,587'Hydroxamate derivatives of selected nonsteroidal antiinflammatory acyl residues and their use for cyclooxygenase and 5-lipoxygenase inhibition'1990 4,939,133'N-substituted-2-hydroxy-.alpha.-oxo-benzeneacetamides and pharmaceutical compositions having activity as modulators of the arachidonic acid cascade'1990 4,931,459'Method for treating acute respirator distress syndrome'1990 4,921,871'Enolamides, pharmaceutical compositions and methods of use thereof for treating inflammation'1990 4,910,317'Benzofurans and benzothiophenes having antiallergic activity and method of use thereof'1990 4,877,881'Process of preparing pyrazoles, isoxazoles and analogs thereof having activity as 5-lipoxygenase inhibitors'1989 4,874,758'Novel enolamides, pharmaceutical compositions and methods of use thereof for activity as modulators of the arachidonic acid cascade'1989 4,868,200'Novel enolamides, pharmaceutical compositions and methods of use thereof for activity as modulators of the arachidonic acid cascade'1989 4,868,205'Novel enolamides, pharmaceutical compositions and methods of use thereof for activity as modulators of the arachidonic acid cascade'1989 4,868,195'Novel enolamides, pharmaceutical compositions and methods of use thereof for activity as modulators of the arachidonic acid cascade'1989 4,868,199'Novel enolamides, pharmaceutical compositions and methods of use thereof for activity as modulators of the arachidonic acid cascade'1989 4,824,958'Process for the preparation of n-1H-tetrazol-5-yl-2-pyrrole carboxamides'1989 4,810,716'Diarylalkanoids having activity as lipoxygenase inhibitors'1989 4,775,677'[3-substituted-2-(substituted imino)-4-oxo-5-thiazolidinylidene]acetic acids having activity as leukotriene antagonists'1988 4,767,776'N-1H-tetrazol-5-yl-2-naphthalene carboxamides and their use as antiallergy and antiinflammatory agents'1988 4,764,525'N-1H-tetrazol-5-ylbenzamides having use as antiallergy and antiinflammatory agents'1988 4,761,424'Enolamides, pharmaceutical compositions and methods for treating inflammation'1988 4,748,183'N-1H-tetrazol-5-yl-2-thiophene carboxamides, N-1H-tetrazol-5-yl-2-pyrrole carboxamides, N-1H-tetrazol-5-yl-2-furan carboxamides, and anti-allergic and anti-inflammatory use thereof'1988 4,703,053'Benzothiophenes and benzofurans and antiallergic use thereof'1987 4,675,332'Acidic tetrazolyl substituted indole compounds and their use as antiallergy agents'1987 4,562,006'Cycloheptadiene derivatives'1985 4,404,138'3-[2-(Azabicyclo) ethyl]-1,2,3,4-tetrahydro-5H-[1]benzopyrano[3,4-c]pyridin-5-ones'1983 4,382,939'3-[2-(Mono-and dialkylamino)propyl]-1,2,3,4-tetrahydro-5H-[1]benzopyrano[3,4-C]pyridin- 5-ones useful for treating bronchospastic diseases'1983 4,360,527'9-(Hydroxy, lower alkoxy or lower alkanoyloxy)-2-(1H-tetrazol-5-yl)naphtho-(2,1-b)-pyran-1-ones and anti-allergic use thereof'1982 4,332,947'Certain 2-pyridylamino-3-thiophene carboxylic acid derivatives'1982 4,287,126'(2-Oxo-2H-1-benzopyran-3-yl)aminooxoacetic acids and their derivatives'1981 4,287,340'Dihydro-oxo-pyrido[1,2-a]thienopyrimidine compounds'1981 4,230,707'Oxo-pyrido[1,2-a]thienopyrimidine compounds and methods for their production'1980 4,225,722'Process for the production of 2-(1H-tetrazol-5-yl)-9-hydroxy-1-oxo-1H-naphtho-(2,1-b) pyran and intermediates therefor'1980 RE030339'Conversion of acid S, produced by the organism Polyangium cellulosum var. fulvum into acid F'1980 4,210,758'1 ,5-Dihydro-1,5-dioxo-N-1H-tetrazol-5-yl-4H-[1]benzopyrano[3,4-b]pyridine- 2-carboxamides'1980 4,198,511'1,5-Dihydro-1,5-dioxo-N- 1H-tetrazol-5-yl-4H-[1]benzopyrano[3,4-b]pyridine-3-carboxamides and process thereof'1980 4,191,825'Diacyloxyacids derived from acid S, an antibiotic produced by Polyangium cellulosum var. fulvum'1980 4,179,447'Process for the production of 2-substituted chromones'1979 4,158,663'Process for the production of 2-substituted chromones'1979 4,138,550'Diacyloxyacids derived from acid S, an antibiotic produced by Polyangium cellulosum var. fulvum'1979 4,127,669'[(4-Oxo-4H-1-benzopyran-3-yl)oxy] acetic acids and derivatives'1978 4,123,536'Dialkyl ({[3-(alkoxycarbonyl)-1,4-dihydro-4-oxo-8-quinolinyl]amino}methylene)pro panedioates'1978 4,117,134'4,5-Dihydro-4,5-dioxo-1H-1-benzopyrano (2,3-B)-pyridine-3-carboxylic acids, salts and esters'1978 4,107,429'1-Nor-2-amino carbamates derived from acid S, an antibiotic produced by Polyangium cellulosum var. fulvum'1978 4,104,274'1-Substituted-2-(2-pyridinyl)ethanone N-oxides'1978 4,098,998'Aldehyde, oxime and phenylhydrazone derivatives of acid S, an antibiotic produced by Polyangium cellulosum var. fulvum'1978 4,076,940'Conversion of acid S, produced by the organism Polyangium cellulosum var. fulvum into acid F'1978 4,076,729'(4-Oxo-4H-1-benzopyran-3-yl)aminooxoacetic acids and their derivatives'1978 4,076,716'Substituted 3-(2-pyridinyl)-4(1H)-quinolinone N-oxides'1978 4,076,720'1-Substituted-2-(2-pyridinyl)ethanone N-oxides'1978 4,066,655'4,10-Dihydro-4,10-dioxo-1H-1-benzopyrano[3,2-b]pyridine-3-carboxylic acids, salts and esters'1978 4,056,532'Alpha-aryl-2-pyridineethanol 1-oxides and alpha-pyridinyl-2-pyridineethanol 1-oxides'1977 4,056,619'1-Substituted-2-(2-pyridinyl)ethanone N-oxides'1977 4,046,769'4,10-Dihydro-4,10-dioxo-1H-1-benzopyrano[3,2-b]pyridine-2-carboxylic acids and esters'1977 4,045,451'2-(Methylthio)naphtho[1,3-bc]pyran-3(2H)-one'1977 4,039,579'2-[1-Imino-2-(methylsulfinyl)ethyl]phenols and 3-[1-imino-2-(methylsulfinyl)ethyl]-2-naphthalenols'1977 4,018,781'2-Aryl substituted isoxazolo(2,3-alpha)pyridinyl halides'1977 4,016,257'Amide derivatives of acids, an antibiotic produced by Polyangium cellulosum var. fulvum'1977 4,013,673'2,3-Dihydro-3-(2-pyridinyl)-4H-1-benzopyran-4-one N-oxides'1977 4,012,422'Process for the cyclization of aryl (methylsulfinyl)-methyl ketones and novel compounds produced thereby'1977 4,009,261'7-Substituted triol derivatives of acid S, an antibiotic produced by polyangium cellulosum var. fulvum'1977 4,007,205'7-Substituted-9-oxoxanthene-2-carboxaldehydes'1977 4,007,193'Substituted 3-(2-pyridinyl)-4(1H)-quinolinone N-oxides'1977 4,001,398'Octahydro and decahydro derivatives of acid S, an antibiotic produced by Polyangium cellulosum var. fulvum'1977 3,983,237'2-Aryl substituted isoxazolo[2,3-a]pyridinyl halides'1976 3,973,020'3-(2-Pyridinyl)-4(1H)-cinnolinone N-oxides'1976 3,932,620'Ketones and ketoximes derived from acid S, an antibiotic produced by polyangium cellulosum var. fulvum'1976 3,932,621'Triols and acetates thereof derived from antibiotic substance, acid S, produced by polyangium cellulosum var. fulvum'1976

Career & activity timeline

Assembled from patent assignee/location history and declaration credentials.

1976–2007Patents assigned to WARNER LAMBERT CO (143)· patent assignee history

1976Patents assigned to VON STRANDTMANN MAX (1)· patent assignee history

1976–1979Based in Parsippany, NJ, US· patent location history

1977Patents assigned to CONNOR DAVID T (1)· patent assignee history

1978–2007Based in Ann Arbor, MI, US· patent location history

2002–2003Patents assigned to MILLENNIUM PHARM INC (4)· patent assignee history

2002Patents assigned to NEUREX CORP (1)· patent assignee history

Inventor activity

Assignee and location history derived from the patent record.

Assignees

Assignee	Patents	Span
WARNER LAMBERT CO	143	1976–2007
MILLENNIUM PHARM INC	4	2002–2003
CONNOR DAVID Tself	1	1977
NEUREX CORP	1	2002
VON STRANDTMANN MAX	1	1976

Locations

Location	Patents	Span
Ann Arbor, MI, US	126	1978–2007
Parsippany, New Jersey, US	25	1976–1979