Inventor
Guenter Linz
Inventor
Mittelbiberach, DE
Overview
Patents· 41 as inventor
Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.
C07Dprimary
C07DHeterocyclic compounds40%
A61PSpecific therapeutic activity of chemical compounds or medicinal preparations30%
C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium12%
A61KPreparations for medical, dental or toiletry purposes11%
C07CAcyclic or carbocyclic compounds7%
PatentTitleYear
9,187,478'Substituted naphthyridines and their use as medicaments'20158,969,568'Substituted naphthyridines and their use as medicaments'20158,933,227'Selective synthesis of functionalized pyrimidines'20158,791,260'Process for the preparation of acylguanidines and acylthioureas'20148,729,265'Regioselective preparation of 2-amino-5-trifluoromethylpyrimidine derivatives'20148,664,222'Specific salt, anhydrous and crystalline form of a dihydropteridione derivative'20148,466,318'Method of preparing chiral cyclic β-aminocarboxamides'20138,372,974'Regioselective preparation of substituted pyrimidines'20138,329,695'Crystalline form of the free base N-[trans-4-[4-(cyclopropylmethyl)-1-piperazinyl]cyclohexyl]-4-[[(7r)-7-ethyl-5,6,7,8-tetrahydro-5-methyl-8-(1-methylethyl)-6-oxo-2-pteridinyl]amino]-3-methoxy-benzamide'20128,304,541'Process for the manufacture of an indolinone derivative'20128,202,867'Methods of using hydrates and polymorphs of 4-[[(7R)-8-cyclopentyl-7-ethyl-5,6,7,8-tetrahydro-5-methyl-6-oxo-2-pteridinyl]amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide'20128,188,086'Specific salt, anhydrous and crystalline form of a dihydropteridione derivative'20128,138,373'Process for the manufacture of dihydropteridinones'20128,138,341'Intermediate compounds useful for the manufacture of dihydropteridinones'2012RE043115'Process for the manufacture of fused piperazin-2-one derivatives'20128,034,816'Hydrates and polymorphs of 4-[[(7R)-8-cyclopentyl-7-ethyl-5,6,7,8-tetrahydro-5-methyl-6-oxo-2-pteridinyl]amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide, process for their manufacture and their use as medicament'20117,759,485'Process for the manufacture of dihydropteridinones'20107,728,134'Hydrates and polymorphs of 4[[(7R)-8-cyclopentyl-7-ethyl-5,6,7,8-tetrahydro-5-methyl-6-oxo-2-pteridinyl]amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide, process for their manufacture and their use as medicament'20107,626,019'Intermediate compounds for the manufacture of fused piperazin-2-one derivatives'20097,514,468'Indolinone derivatives substituted in the 6 position, the preparation thereof and their use as pharmaceutical compositions'20097,439,358'Specific salt, anhydrous and crystalline form of a dihydropteridione derivative'20087,294,721'(R)-2-(4-amidinophenylaminomethyl)-1-methyl-5-[1-(carboxymethylamino)-1(pyrrolidinocarbonyl)-ethyl]-benzimidazole, the monohydrochloride thereof, preparation thereof and the use as pharmaceutical composition'20077,238,807'Process for the manufacture of fused piperazin-2-one derivatives'20077,169,934'(R) 2-(4-amidinophenylaminomethyl)-1-methyl-5-[1-(carboxymethylamino)-1 (pyrrolidinocarbonyl)-ethyl]-benzimidazole, the monohydrochloride thereof, preparation thereof and the use as pharmaceutical composition'20077,119,093'3-Z-[1-(4-(N-((4-Methyl-piperazin-1-yl)-methylcarbonyl)-N-methyl-amino)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone-monoethanesulphonate and the use thereof as a pharmaceutical composition'20066,919,325'Pharmaceutical compositions containing tiotropium salts and low-solubility salmeterol salts'20056,756,508'Cinnamic acid salts, processes for their preparation, and their use as medicaments'20046,680,345'Salicylic acid salts of salmeterol'20045,852,192'Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them'19985,650,424'Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them'19975,591,769'Cyclic imino derivatives and pharmaceutical compositions containing them'19975,576,444'Cyclic imino derivatives, processes for preparing them and pharmaceutical compositions containing these compounds'19965,563,268'Heterobiaryl derivatives'19965,541,343'Cyclic imino derivatives and pharmaceutical compositions containing them'19965,489,693'Cyclic imino derivatives, pharmaceutical compositions containing these compounds and processes preparing them'19965,478,942'Cyclic urea derivatives and pharmaceutical compositions containing these compounds'19955,463,071'5-membered heterocyclic compounds, processes for preparing them and pharmaceutical compositions containing these compounds'19955,455,348'2-pyrrolidinones, pharmaceutical compositions containing these compounds and processes for preparing them'19955,434,150'Condensed 5-membered heterocyclic compounds, processes for preparing them and pharmaceutical preparations containing these compounds'19955,418,233'Heterobiarly derivatives and pharmaceutical compositions thereof'19955,276,049'Cyclic urea derivatives, pharmaceutical compositions containing these compounds and methods of using the same'1994Career & activity timeline
Assembled from patent assignee/location history and declaration credentials.
1994–1998Patents assigned to THOMAE GMBH DR K (12)· patent assignee history
1994–2015Based in Mittelbiberach, DE· patent location history
1995Based in Mittelberach, DE· patent location history
2004–2015Patents assigned to BOEHRINGER INGELHEIM PHARMA (7)· patent assignee history
2007–2015Patents assigned to BOEHRINGER INGELHEIM INT (21)· patent assignee history
2012–2015Patents assigned to LINZ GUENTER (14)· patent assignee history
2012–2015Patents assigned to KRAEMER GERD (6)· patent assignee history
Inventor activity
Assignee and location history derived from the patent record.
Assignees
| Assignee | Patents | Span |
|---|---|---|
| BOEHRINGER INGELHEIM INT | 21 | 2007–2015 |
| LINZ GUENTERself | 14 | 2012–2015 |
| THOMAE GMBH DR K | 12 | 1994–1998 |
| BOEHRINGER INGELHEIM PHARMA | 7 | 2004–2015 |
| KRAEMER GERD | 6 | 2012–2015 |
Locations
| Location | Patents | Span |
|---|---|---|
| Mittelbiberach, DE | 40 | 1994–2015 |
| Mittelberach, DE | 1 | 1995 |