Inventor

Richard B. Sparks

Inventor
Wilmington, DE, US

Overview

62→
Patents
1997–2021
Patent span
Human necessities
Primary field (CPC A)

Patents· 62 as inventor

Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.

C07Dprimary
C07DHeterocyclic compounds39%
A61PSpecific therapeutic activity of chemical compounds or medicinal preparations37%
A61KPreparations for medical, dental or toiletry purposes20%
C07BGeneral methods of organic chemistry2%
C07CAcyclic or carbocyclic compounds2%
C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium1%
PatentTitleYear
11,091,491Heterocyclic compounds as PI3K-y inhibitors202110,738,057Tertiary alcohols as PI3K-g inhibitors202010,653,6771,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase202010,646,492Heterocyclylamines as PI3K inhibitors202010,618,910Tricyclic heterocycles as BET protein inhibitors202010,479,795Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines and substituted imidazo[1,2-b]pyridazines as PI3K-gamma inhibitors201910,472,368Heterocyclic compounds as PI3K-g inhibitors201910,464,947Tricyclic heterocycles as BET protein inhibitors201910,376,513Heterocyclylamines as PI3K inhibitors201910,369,1371,2,5-Oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase201910,259,818Bicyclic azaheterocyclobenzylamines as PI3K inhibitors201910,227,359Tricyclic heterocycles as bet protein inhibitors201910,138,248Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines, substituted imidazo[1,2-b]pyridazines and substituted imidazo[1,2-a]pyrazines as PI3K-g inhibitors201810,092,570Heterocyclylamines as PI3K inhibitors201810,034,8641,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase20189,944,646Bicyclic azaheterocyclobenzylamines as PI3K inhibitors20189,938,294Tricyclic heterocycles as BET protein inhibitors20189,879,010'Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b] pyrimidin-5-yl-amines as Janus kinase inhibitors'20189,834,565Tricyclic heterocycles as bet protein inhibitors20179,815,839'N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors'20179,789,094'1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase'20179,730,939'Heterocyclylamines as PI3K inhibitors'20179,624,241'Tricyclic heterocycles as BET protein inhibitors'20179,580,419'Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors'20179,527,864'Tricyclic heterocycles as BET protein inhibitors'20169,527,848'N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors'20169,403,847'Substituted heteroaryl fused derivatives as P13K inhibitors'20169,320,732'1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase'20169,309,251'Bicyclic azaheterocyclobenzylamines as PI3K inhibitors'20169,290,514'Tricyclic heterocycles as BET protein inhibitors'20169,227,985'Tricyclic heterocycles as bet protein inhibitors'20169,193,721'Fused derivatives as PI3Kδ inhibitors'20159,096,600'N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors'20159,090,611'Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as janus kinase inhibitors'20158,993,605'1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase'20158,951,536'N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase'20158,871,753'Macrocyclic compounds and their use as kinase inhibitors'20148,835,423'Azepine inhibitors of janus kinases'20148,822,511'1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase'20148,796,319'1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase'20148,765,727'Macrocyclic compounds and their use as kinase inhibitors'20148,759,359'Substituted heteroaryl fused derivatives as PI3K inhibitors'20148,741,895'Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors'20148,563,541'Azepine inhibitors of Janus kinases'20138,507,541'N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase'20138,450,351'N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase'20138,445,488'Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors'20138,377,976'N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase'20138,088,803'1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase'20128,053,433'Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as janus kinase inhibitors'20117,335,667'Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-4-yl-amines as Janus kinase inhibitors'20087,141,596'Inhibitors of proteins that bind phosphorylated molecules'20066,737,424'Alpha-substituted pyridazino quinoline compounds'20046,232,313'Pyridazino quinoline compounds'20016,214,826'Pyridazino quinoline compounds'20016,103,721'Heteroaryl-substituted pyridazino quinoline compounds'20005,837,705'Alpha-substituted pyridazino quinoline compounds'19985,744,471'Pyridazion quinoline compounds'19985,739,133'Pyridazinedione compounds useful in treating neurological disorders'19985,733,910'Pyridazinedione compounds useful in the treating neurological disorders'19985,604,227'Pyridazinedione compounds useful in treating neurological disorders'19975,599,814'Pyridazinedione compounds useful in treating neurological disorders'1997

Career & activity timeline

Assembled from patent assignee/location history and declaration credentials.

1997–2004Based in Linwood, PA, US· patent location history
1998–2004Patents assigned to ZENECA LTD (7)· patent assignee history
2001–2014Based in Boothwyn, PA, US· patent location history
2006–2021Patents assigned to INCYTE CORP (52)· patent assignee history
2012–2015Patents assigned to SPARKS RICHARD B (12)· patent assignee history
2012–2015Patents assigned to COMBS ANDREW P (10)· patent assignee history
2013–2020Based in Wilmington, DE, US· patent location history
2015–2020Patents assigned to INCYTE HOLDINGS CORP (23)· patent assignee history
2019–2021Based in Hockessin, DE, US· patent location history

Inventor activity

Assignee and location history derived from the patent record.

Assignees
AssigneePatentsSpan
INCYTE CORP522006–2021
INCYTE HOLDINGS CORP232015–2020
SPARKS RICHARD Bself122012–2015
COMBS ANDREW P102012–2015
ZENECA LTD71998–2004
Locations
LocationPatentsSpan
Wilmington, Delaware, US382013–2020
Boothwyn, Pennsylvania, US132001–2014
Linwood, Pennsylvania, US91997–2004
Hockessin, Delaware, US22019–2021