Inventor
Andreas Maderna
Inventor
Stony Point, NY, US
Overview
Patents· 23 as inventor
Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.
C07Dprimary
C07DHeterocyclic compounds25%
A61PSpecific therapeutic activity of chemical compounds or medicinal preparations24%
A61KPreparations for medical, dental or toiletry purposes18%
C07CAcyclic or carbocyclic compounds8%
C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium8%
C07KPeptides8%
C07BGeneral methods of organic chemistry5%
C07HSugars5%
Y02ATechnologies for adaptation to climate change1%
PatentTitleYear
10,968,242Cyclopentane-based modulators of STING (stimulator of interferon genes)202110,870,706Bifunctional cytotoxic agents containing the CTI pharmacophore202010,662,204Substituted quinazoline and pyridopyrimidine derivatives useful as anticancer agents202010,590,115Tetrahydroquinazoline derivatives useful as anticancer agents202010,544,0953-indol substituted derivatives, pharmaceutical compositions and methods for use202010,538,542Cyclopentane-based modulators of STING (stimulator of interferon genes)202010,391,182Bifunctional cytotoxic agents201910,086,085Bifunctional cytotoxic agents20189,873,6903-indol substituted derivatives, pharmaceutical compositions and methods for use20189,296,686'Preparation of (R)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide and (S)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide'20169,249,186'Cytotoxic peptides and antibody drug conjugates thereof'20169,138,486'Cytotoxic peptides and antibody drug conjugates thereof'20158,884,058'Preparation of (R)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide and (S)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide'20148,828,401'Cytotoxic peptides and antibody drug conjugates thereof'20148,829,052'Derivatives of N-(arylamino)sulfonamides as inhibitors of MEK'20148,513,443'Preparation of (R)-N-(3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide and (S)-N-3,4-difluoro-2(2-fluoro-4-iodophenylamino)-6-methoxyphenyl)-1-(2,3-dihydroxypropyl)cyclopropane-1-sulfonamide'20138,101,799'Derivatives of N-(arylamino) sulfonamides as inhibitors of MEK'20128,063,049'Inhibitors of MEK'20117,820,664'Inhibitors of MEK'20107,759,518'Derivatives of N-(arylamino) sulfonamides as inhibitors of MEK'20107,652,047'Phenylamino isothiazole carboxamidines as MEK inhibitors'20107,429,667'Phenylamino isothiazole carboxamidines as MEK inhibitors'20086,664,426'Ether and ester derivatives of the perborate icosahedron'2003Career & activity timeline
Assembled from patent assignee/location history and declaration credentials.
2003–2010Based in Los Angeles, CA, US· patent location history
2008–2016Patents assigned to ARDEA BIOSCIENCES INC (8)· patent assignee history
2010–2014Patents assigned to ARDEA BIOSCIENCES (3)· patent assignee history
2010–2018Based in Stony Point, NY, US· patent location history
2011–2014Patents assigned to MADERNA ANDREAS (4)· patent assignee history
2011–2014Patents assigned to VERNIER JEAN-MICHEL (4)· patent assignee history
2014–2021Patents assigned to PFIZER (12)· patent assignee history
2019–2020Based in Escondido, CA, US· patent location history
2020Based in San Diego, CA, US· patent location history
2021Based in Walnut Creek, CA, US· patent location history
Inventor activity
Assignee and location history derived from the patent record.
Assignees
| Assignee | Patents | Span |
|---|---|---|
| PFIZER | 12 | 2014–2021 |
| ARDEA BIOSCIENCES INC | 8 | 2008–2016 |
| MADERNA ANDREASself | 4 | 2011–2014 |
| VERNIER JEAN-MICHEL | 4 | 2011–2014 |
| ARDEA BIOSCIENCES | 3 | 2010–2014 |
Locations
| Location | Patents | Span |
|---|---|---|
| Stony Point, New York, US | 13 | 2010–2018 |
| Escondido, California, US | 4 | 2019–2020 |
| Los Angeles, California, US | 3 | 2003–2010 |
| San Diego, California, US | 2 | 2020 |
| Walnut Creek, California, US | 1 | 2021 |