Inventor
George D. Maynard
Inventor
Clinton, CT, US
Overview
Patents· 65 as inventor
Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.
C07Dprimary
C07DHeterocyclic compounds49%
A61PSpecific therapeutic activity of chemical compounds or medicinal preparations35%
A61KPreparations for medical, dental or toiletry purposes7%
C07BGeneral methods of organic chemistry2%
G01NInvestigating or analysing materials by determining their chemical or physical properties2%
Y10STechnical subjects covered by former uspc cross-reference art collections [xracs] and digests2%
C07CAcyclic or carbocyclic compounds1%
C40BCombinatorial chemistry1%
PatentTitleYear
8,633,193'Pyrrolo-pyridine, pyrrolo-pyrimidine and related heterocyclic compounds'20148,338,591'3-aryl-5,6-disubstituted pyridazines'20128,129,395'4,5-disubstituted-2-aryl pyrimidines'20128,119,665'Aryl imidazoles and related compounds as C5a receptor modulators'20127,915,288'1-aryl-4-substituted isoquinolines'20117,906,528'Pyrrolo-pyridine, pyrrolo-pyrimidine and related heterocyclic compounds'20117,863,454'3-substituted-6-aryl pyridines'20117,642,267'Benzimidazole and pyridylimidazole derivatives'20107,482,350'4,5-disubstituted-2-aryl pyrimidines'20097,342,115'3-substituted-6-aryl pyridines'20087,300,945'Benzimidazole and pyridylimidazole derivatives'20077,282,498'Substituted fused pyrroleoximes and fused pyrazoleoximes'20077,271,170'Imidazo-pyrimidines and triazolo-pyrimidines: benzodiazepine receptor ligands'20077,186,734'Aryl imidazoles and related compounds as C5a receptor modulators'20077,122,546'Imidazol-1-ylmethyl pyridazine derivatives'20067,041,664'2-aminoquinolinecarboxamides: neurokinin receptor ligands'20067,037,922'Aryl fused 2,4-disubstituted pyridines: NK3 receptor ligands'20067,030,144'Substituted imidazole derivatives: GABAA receptor ligands'20066,982,268'Substituted imidazolylmethyl pyridine and pyrazine derivatives GABAA receptor ligands'20066,951,864'4-imidazol-1-ylmethyl-pyrimidine derivatives'20056,949,562'Heterocyclic compounds as ligands of the GABAA receptor'20056,936,617'Heteroaryl substituted fused bicyclic heteroaryl compound as GABAA receptor ligands'20056,916,827'Substituted ring-fused imidazole derivative: GABAA receptors ligands'20056,916,819'Benzimidazole and pyridylimidazole derivatives'20056,894,044'2-aminoquinolinecarboxamides: neurokinin receptor ligands'20056,884,815'High affinity small molecule C5a receptor modulators'20056,861,529'Cycloalkypyrrole-3-carboxylic acid derivatives and heterocycloalkylpyrrole-3-carboxylic acid derivatives'20056,852,730'Substituted fused pyrazolecarboxylic acid arylamides and related compounds'20056,743,817'Substituted fused pyrroleimines and pyrazoleimines'20046,723,743'High affinity small molecule C5a receptor modulators'20046,673,811'1H-pyrrolo 3,2-b pyridine-3-carboxylic acid amines as GABAA receptor ligands'20046,656,941'Aryl substituted tetrahydroindazoles'20036,653,471'Heterocyclic compounds as ligands of the GABAA receptor'20036,624,175'4-Substituted quinoline derivatives'20036,509,366'Substituted imidazoles as selective modulators of Bradykinin B2 receptors'20036,472,402'Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino 2,3-Bindole derivatives'20026,423,704'Substituted 4-(1H-benzimidazol-2-yl)1,4diazepanes useful for the treatment of allergic diseases'20026,420,365'Imidazopyridines and related derivatives as selective modulators of bradykinin B2 receptors'20026,413,982'4-substituted quinoline derivatives'20026,369,053'2-Aminoquinolinecarboxamides: neurokinin receptor ligands'20026,362,186'Aminoalkyl substituted 9H-phridino2,3-b indole and 9H-pyrimidino4,5-b indole derivatives'20026,358,949'Aryl and hetroaryl fused aminoalkyl-imidazole derivatives: selective modulators of bradykinin B2 receptors'20026,316,445'Carboxy substituted acylic carboxamide derivatives'20016,291,473'Aminoalkyl substituted 5,6,7,8-tetrahydro-9H-pyridino [2, 3-B] indole and 5,6,7,8-tetrahydro-9H-pyrimidino [4, 5-B] indole derivatives: CRF1 specific ligands'20016,221,875'Substituted 9H-pyridino [2,3-B]indole and 9H-pyrimidino [4,5-B]indole derivatives: selective neuropeptide Y receptor ligands'20016,211,199'Substituted 4-(1H-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseases'20016,194,406'Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic disease'20016,147,085'Aminoalkyl substituted 9H-pyridino[2,3-b] indole and 9H-pyrimidino[4,5-b] indole derivatives'20005,977,139'Carboxysubstituted cyclic carboxamide derivatives'19995,932,571'Substituted N-methyl-N-(4-(4-(1H-benzimidazol-2-yl) {1,4}diazepan-1-yl)-2-(aryl) butyl) benzamides useful for the treatment of allergic diseases'19995,922,737'Substituted N-methyl-N-(4-(4-(1H-Benzimidazol-2-YL-amino) piperidin-1-YL)-2-(arlyl) butyl) benzamides useful for the treatment of allergic diseases'19995,861,417'Heterocyclic substituted pyrrolidine amide derivatives'19995,861,416'Substituted pyrrolidin-3-yl-alkyl-piperidines'19995,824,690'Substituted pyrrolidin-3-yl-alkyl-piperidines'19985,739,150'Piperidinyl thiacyclic derivatives'19985,661,160'Substituted pyrrolidin-3-yl-alkyl-piperidines'19975,650,416'Piperidinyl thiacyclic derivatives'19975,648,366'Substituted pyrrolidin-3-yl-alkyl-piperidines'19975,635,510'Substituted pyrrolidin-3-yl-alkyl-piperidines'19975,631,268'Piperidinyl thiacyclic derivatives'19975,602,147'Piperidinyl thiacyclic derivatives'19975,596,003'Piperidinyl thiacyclic derivatives'19975,541,200'Piperidinyl thiacyclic derivatives'19965,476,861'Piperidinyl thiacyclic derivatives'19955,371,093'Piperidinyl thiacyclic derivatives'1994Career & activity timeline
Assembled from patent assignee/location history and declaration credentials.
1994–1999Based in Cincinnati, OH, US· patent location history
1996–1999Patents assigned to MERRELL PHARMA INC (10)· patent assignee history
1998–1999Patents assigned to HOECHST MARION ROUSSEL INC (5)· patent assignee history
1999–2001Based in Westbrook, CT, US· patent location history
2000–2010Patents assigned to NEUROGEN CORP (36)· patent assignee history
2000–2014Based in Clinton, CT, US· patent location history
2001–2002Patents assigned to AVENTIS PHARMA INC (4)· patent assignee history
2011–2012Patents assigned to NOVARTIS INT PHARM LTD (6)· patent assignee history
Inventor activity
Assignee and location history derived from the patent record.
Assignees
| Assignee | Patents | Span |
|---|---|---|
| NEUROGEN CORP | 36 | 2000–2010 |
| MERRELL PHARMA INC | 10 | 1996–1999 |
| NOVARTIS INT PHARM LTD | 6 | 2011–2012 |
| HOECHST MARION ROUSSEL INC | 5 | 1998–1999 |
| AVENTIS PHARMA INC | 4 | 2001–2002 |
Locations
| Location | Patents | Span |
|---|---|---|
| Clinton, CT, US | 46 | 2000–2014 |
| Cincinnati, OH, US | 14 | 1994–1999 |
| Westbrook, CT, US | 5 | 1999–2001 |