Inventor

Bernward Scholkens

Inventor

Kelkheim, DE

Overview

1977–2008

Patent span

Human necessities

Primary field (CPC A)

Patents· 57 as inventor

Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.

A61Pprimary

A61PSpecific therapeutic activity of chemical compounds or medicinal preparations27%

C07DHeterocyclic compounds24%

A61KPreparations for medical, dental or toiletry purposes23%

C07KPeptides15%

C07CAcyclic or carbocyclic compounds7%

Y10STechnical subjects covered by former uspc cross-reference art collections [xracs] and digests2%

Y02PClimate change mitigation technologies in the production or processing of goods1%

C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium1%

C07HSugars1%

PatentTitleYear

7,368,469'Use of inhibitors of the renin-angiotensin system in the prevention of cardiovascular events'2008 6,462,024'Use of inhibitors of the sodium-hydrogen exchanger for the production of a medicament for decreasing undesired effects of substrates of the heart'2002 6,211,196'Benzyloxy-substituted, fused N-heterocycles, processes for their preparation, and their use as bradykinin receptor antagonists'2001 6,140,341'Aminoalkyl and acylaminoalkyl ethers, process for their preparation, and their use as bradykinin receptor antagonists'2000 5,859,025'Fluoroalkyl- and fluoroalkoxy-substituted heterocyclic bradykinin antagonists, process for their preparation, and their use'1999 5,834,500'Sulfur-containing heterocyclic bradykinin antagonists, process for their preparation, and their use'1998 5,747,504'Method of treating cardiac insufficiency using angiotensin-converting enzyme inhibitors'1998 5,744,496'Method of treating cardiac insufficiency using angiotensin-converting enzyme inhibitors'1998 5,739,300'Antiadhesive piperidine-and pyrrolidinecarboxylic acids'1998 5,684,016'Method of treating cardiac insufficiency'1997 5,648,333'Peptides having bradykinin antagonist action'1997 5,635,525'Benzimidazole derivatives as angiotensin II receptor antagonists, pharmacticals, and treatment of hypertension therewith'1997 5,597,803'Bradykinin peptides with modifications at the N terminus'1997 5,482,957'Azole derivatives, process for their preparation and their use'1996 5,444,068'Imidazopyridine derivatives as angiotensin II receptor antagonists, pharmaceuticals, and treatment of hypertension therewith'1995 5,440,046'Substituted imidazoles'1995 5,403,856'Method of treating cardiac insufficiency using angiotensin-converting enzyme inhibitors'1995 5,401,766'Aminoacid derivatives, a process for their preparation, agents containing these compounds, and the use thereof'1995 5,364,878'Use of substituted 3,4-dihydro-2H-benzopyrans as remedies for obstructive functional disorders of the lungs'1994 5,360,791'Renin-inhibiting aminodiol derivatives'1994 5,350,751'Substituted imidazoles, pharmaceutical compositions containing these, and the use thereof as antagonists of angiotensin II receptors for the treatment of high blood pressure'1994 5,292,755'USPA benzolyguanidines'1994 5,236,943'Method for the treatment of cardiac and of vascular hypertrophy and hyperplasia'1993 5,231,080'Method for the treatment of atherosclerosis, thrombosis, and peripheral vessel disease'1993 5,231,083'Method for the treatment of cardiac and of vascular hypertrophy and hyperplasia'1993 5,225,414'Substituted azoles, a process for their preparation, and their use'1993 5,215,968'Dipeptide derivatives having an enzyme inhibitory action'1993 5,204,357'Renin-inhibiting amino acid derivatives'1993 5,194,442'2,3,4,5-tetrahydro-1-benzoxepins, the use thereof and pharmaceutical products based on these compounds'1993 5,185,324'Enzyme-inhibiting amino acid derivatives, a process for the preparation thereof, agents containing these, and the use thereof'1993 5,169,841'Renin inhibitors'1992 5,162,362'Octahydroindole-2-carboxylic acids'1992 5,158,959'Decahydroisoquinoline carboxylic acids'1992 5,130,310'Substituted benzo[b]pyrans, processes for their preparation, their use and pharmaceutical preparations based on these compounds'1992 5,116,835'Enzyme-inhibiting urea derivatives of dipeptides, a process for the preparation thereof, agents containing these, and the use thereof'1992 5,091,394'Benzoylguanidines, a process for their preparation, their use as medicaments and medicaments containing them'1992 5,061,722'Cis, endo-2-azabicyclo-[3.3.0]-octane-3-carboxylic acids, a process for their preparation, agents containing these compounds and their use'1991 5,053,519'Cis, endo-2-azabicyclo-[3.3.0]-octane-5-carboxylic acids'1991 5,043,344'Unsaturated N-benzopyranyllactams'1991 5,025,010'Benzothiazinone derivatives, and pharmaceuticals containing them'1991 4,999,371'Substituted 3,4-dihydro-2H-benzopyrans, processes for their preparation, their use and pharmaceutical products based on these compounds'1991 4,879,403'Process for the preparation of cis, endo-2-azabicyclo-[3.3.0]-octane-3-carboxylic acids'1989 4,861,755'Peptides with vasorelaxant, natriuretic and diuretic effects a process for their preparation, agents containing them, and their use'1989 4,857,520'Fused azepinone and azocinone derivatives, processes for their preparation, agents containing them and their use, and intermediates in their preparation'1989 4,855,286'Renin-inhibiting di- and tripeptides, a process for their preparation, agents containing them, and their use'1989 4,727,160'Method for making 2-azabicyclo-[3.3.0]-octane-3-carboxylic acids'1988 4,624,962'Substituted derivatives of 2-azabicyclo-[3.3.0]octanes'1986 4,595,675'Bicyclic .alpha.-iminocarboxylic acid compounds having hypotensive activity'1986 4,515,803'Substituted derivatives of octahydroindole-2-carboxylic acids'1985 4,371,542'Hetero-imino-prostacyclins'1983 4,312,882'Thienyoxy and furyl containing analogs of prostacyclin and their use as medicaments'1982 4,304,783'Thienyl, thienyloxy or furyl substituted prostaglandin derivatives in the 6-keto-PGE.sub.1 series'1981 4,198,429'Esters of 5-methyl-10,11-dihydroprostaglandin-A.sub.1'1980 4,182,773'Novel prostaglandin derivatives'1980 4,079,145'Certain pyrrolidone derivatives and pharmaceutical use thereof'1978 4,061,766'Cyclopentane derivatives and process for preparing them'1977 4,013,791'Peptides having an antihypertensive effect'1977

Career & activity timeline

Assembled from patent assignee/location history and declaration credentials.

1977–2000Patents assigned to HOECHST AG (54)· patent assignee history

1977–2008Based in Kelkheim, DE· patent location history

1977Based in Bad Soden, DE· patent location history

1993–1997Based in Taunus, DE· patent location history

1995Based in Kelheim/Donau, DE· patent location history

2001–2002Patents assigned to AVENTIS PHARMA GMBH (2)· patent assignee history

2008Patents assigned to SANOFI AVENTIS DEUTSCHLAND (1)· patent assignee history

Inventor activity

Assignee and location history derived from the patent record.

Assignees

Assignee	Patents	Span
HOECHST AG	54	1977–2000
AVENTIS PHARMA GMBH	2	2001–2002
SANOFI AVENTIS DEUTSCHLAND	1	2008

Locations

Location	Patents	Span
Kelkheim, DE	53	1977–2008
Taunus, DE	2	1993–1997
Kelheim/Donau, DE	1	1995
Bad Soden, DE	1	1977