Inventor

Michelangelo Scalone

Inventor

Birsfelden, CH

Overview

1992–2021

Patent span

Chemistry

Primary field (CPC C)

Patents· 54 as inventor

Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.

C07Dprimary

C07DHeterocyclic compounds29%

A61PSpecific therapeutic activity of chemical compounds or medicinal preparations16%

C07CAcyclic or carbocyclic compounds13%

C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium10%

Y02PClimate change mitigation technologies in the production or processing of goods8%

A61KPreparations for medical, dental or toiletry purposes7%

C07BGeneral methods of organic chemistry7%

B01JChemical or physical processes, e.g. catalysis or colloid chemistry6%

C12PFermentation or enzyme-using processes to synthesise a desired chemical compound or composition or to separate optical isomers from a racemic mixture2%

C07JSteroids1%

PatentTitleYear

11,124,532Chiral metal complex compounds2021 10,858,324Processes for the preparation of pyrimidinylcyclopentane compounds2020 10,435,378Processes for the preparation of pyrimidinylcyclopentane compounds2019 10,329,288Process for preparing a compound2019 9,862,689'Processes for the preparation of pyrimidinylcyclopentane compounds'2018 9,603,816'Process'2017 9,562,009'Process to manufacture N-[(3S)-1-[4-[(3-fluorophenyl)methoxy]phenyl]-5-oxo-pyrrolidin-3-yl]acetamide'2017 9,353,081'Bicyclic dihydroquinoline-2-one derivatives'2016 8,975,438'Process for the preparation of cyclohexanecarboxylic acid derivatives'2015 8,664,403'Process'2014 8,450,496'Process for the preparation of propionic acid derivatives'2013 8,288,534'Process for the preparation a ruthenium complex'2012 8,106,187'Process for the preparation of a macrocycle'2012 7,939,668'Ruthenium complexes as catalysts for metathesis reactions'2011 7,910,728'Process for the preparation of a macrocycle'2011 7,781,586'Metathesis catalysts'2010 7,772,264'Salt and polymorphs of a DPPIV inhibitor'2010 7,691,876'Heterobicyclic amide compounds'2010 7,642,366'Phosphine ligands'2010 7,365,207'Process for the production of chiral propionic acid derivatives'2008 7,262,303'Process for the production of chiral propionic acid derivatives'2007 7,259,176'Process for the preparation of the insulin sensitizer'2007 7,238,816'Preparation of epothilone derivatives'2007 7,169,935'Process for preparing heterocyclic indene analogs'2007 6,914,140'Asymmetric synthesis process'2005 6,858,749'Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-one'2005 6,818,774'Isoquinoline derivatives'2004 6,818,789'Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-one'2004 6,777,559'Process for preparing heterocyclic indene analogs'2004 6,753,432'Process for the preparation of thiazolidinedione derivatives'2004 6,743,927'Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-one'2004 6,620,941'Process for the preparation of thiazolidinedione derivatives'2003 6,605,723'Process for the preparation of ethanesul fonyl-piperidine derivatives'2003 6,552,204'Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-one'2003 6,545,165'Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-one'2003 6,531,597'Process for preparation of 2-phenyl acetic acid derivatives'2003 6,531,609'Process for the preparation of thiazolidinedione derivatives'2003 6,482,958'Methods for the preparation of 4-hydroxy benzothiophene'2002 6,437,118'Vinylating of pyrimidine derivatives'2002 6,437,144'Methods for the preparation of 4-hydroxy benzothiophene'2002 6,348,612'Chiral amido-phosphine-phosphinite compounds'2002 6,300,509'Amino-amide-ruthenium complexes'2001 6,291,685'Methods for the preparation of 4-hydroxybenzothiophene'2001 6,277,997'Process for the preparation of chiral lactones'2001 6,222,039'Process for the preparation of chiral lactones'2001 6,187,961'Process for the preparation of trans-(R,R)-actinol'2001 6,069,245'Asymmetric synthesis of azepines'2000 5,902,882'Assymetric synthesis of azepines'1999 5,880,285'Process for manufacture of optically active isochinole compounds'1999 5,534,635'Process for preparing pyridine-2-carboxamides'1996 5,393,900'Steroid intermediates for the formation of vitamin D.sub.3 analogues'1995 5,380,861'Process for preparing pyridine 2-carboxamides'1995 5,342,833'Vitamin D3 analogs'1994 5,110,955'Tocopherol synthesis: chromane cyclization and catalysis'1992

Career & activity timeline

Assembled from patent assignee/location history and declaration credentials.

1992–2021Patents assigned to HOFFMANN LA ROCHE (37)· patent assignee history

1992–2020Based in Birsfelden, CH· patent location history

2003–2005Patents assigned to ROCHE COLORADO CORP (5)· patent assignee history

2010Based in Baslerstrasse, CH· patent location history

2011–2012Patents assigned to ROCHE PALO ALTO LLC (4)· patent assignee history

2012–2016Patents assigned to SCALONE MICHELANGELO (6)· patent assignee history

2018–2020Patents assigned to GENENTECH INC (4)· patent assignee history

2021Based in Basel, CH· patent location history

Inventor activity

Assignee and location history derived from the patent record.

Assignees

Assignee	Patents	Span
HOFFMANN LA ROCHE	37	1992–2021
SCALONE MICHELANGELOself	6	2012–2016
ROCHE COLORADO CORP	5	2003–2005
GENENTECH INC	4	2018–2020
ROCHE PALO ALTO LLC	4	2011–2012

Locations

Location	Patents	Span
Birsfelden, CH	52	1992–2020
Basel, CH	1	2021
Baslerstrasse, CH	1	2010