Inventor
Frank Kayser
Inventor
San Francisco, CA, US
Overview
Patents· 43 as inventor
Public. Assignee & technology derived from the patent record. Each patent links to its LexDana page.
C07Dprimary
C07DHeterocyclic compounds33%
A61PSpecific therapeutic activity of chemical compounds or medicinal preparations25%
A61KPreparations for medical, dental or toiletry purposes16%
C07CAcyclic or carbocyclic compounds12%
C07FAcyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium8%
C07BGeneral methods of organic chemistry6%
C12NMicroorganisms or enzymes1%
PatentTitleYear
11,046,680Heteroaryl-substituted triazoles as APJ receptor agonists202110,736,883Triazole furan compounds as agonists of the APJ receptor202010,562,857Ion channel inhibitory compounds, pharmaceutical formulations, and uses202010,221,162Triazole agonists of the APJ receptor20199,868,721'Triazole agonists of the APJ receptor'20189,850,183Conjugates derived from non-steroidal anti-inflammatory drugs and methods of use thereof in imaging20179,745,286'Triazole agonists of the APJ receptor'20179,656,997'Triazole agonists of the APJ receptor'20179,593,129'Piperidinone derivatives as MDM2 inhibitors for the treatment of cancer'20179,573,936'Triazole agonists of the APJ receptor'20179,376,425'Heterocyclic compounds as MDM2 inhibitors for the treatment of cancer'20169,296,736'Piperidinone derivatives as MDM2 inhibitors for the treatment of cancer'20168,426,358'Methods for treating atherosclerosis'20137,776,867'Furanopyrimidines'20107,763,624'Substituted pyrazolo[3,4-d]pyrimidines as ACK-1 and LCK inhibitors'20107,674,907'Furanopyridine derivatives and methods of use'20107,645,779'Linked biaryl compounds'20107,511,043'FXR modulators'20097,473,703'Heterocyclic arylsulfonamidobenzylic compounds'20097,358,250'Pyrrolo[2,3-d]pyrimidines that modulate ACK1 activity'20087,326,812'Arylsulfonamidobenzylic compounds'20087,300,932'Pyrrolo[1,2-b]pyridazine derivatives'20077,244,727'Fused bicyclic nitrogen-containing heterocycles'20077,112,606'Heterocyclic arylsulfonamidobenzylic compounds'20067,071,358'Arylsulfonamidobenzylic compounds'20066,869,975'Linked biaryl compounds'20056,777,446'FXR modulators'20046,632,836'Carbocyclic potassium channel inhibitors'20036,455,548'4-alkyl piperidinyl pyrrolidine modulators of chemokine receptor activity'20026,303,637'Heterocyclic potassium channel inhibitors'20016,303,593'3-thienyl and 3-furanyl pyrrolidine modulators of chemokine receptor activity'20016,194,458'Benzamide potassium channel inhibitors'20016,100,293'Tetracyclic triterpene derivatives with immunosuppressant activity'20006,083,980'Furanyl, tetracyclic triterpene derivatives with immunosuppressant activity'20006,051,590'Immunosuppressant tricyclic compounds'20006,022,890'Immunosuppressant tetracyclic triterpenes'20005,998,408'Triterpene derivatives with immunosuppressant activity'19995,952,371'Triterpene derivatives with immunosuppressant activity'19995,883,119'Triterpene derivatives with immunosuppressant activity'19995,874,594'Triterpene derivatives with immunosuppressant activity'19995,763,478'Triterpene derivatives with immunosuppressant activity'19985,696,156'Triterpene derivatives with immunosuppressant activity'19975,679,705'Triterpene derivatives with immunosuppressant activity'1997Career & activity timeline
Assembled from patent assignee/location history and declaration credentials.
1997–2003Patents assigned to MERCK & CO INC (16)· patent assignee history
1997–2003Based in Hoboken, NJ, US· patent location history
2001–2021Based in San Francisco, CA, US· patent location history
2004–2005Patents assigned to TULARIK INC (2)· patent assignee history
2005–2010Patents assigned to JAPAN TOBACCO INC (4)· patent assignee history
2006–2021Patents assigned to AMGEN INC (21)· patent assignee history
2020Patents assigned to AFASCI INC (1)· patent assignee history
Inventor activity
Assignee and location history derived from the patent record.
Assignees
| Assignee | Patents | Span |
|---|---|---|
| AMGEN INC | 21 | 2006–2021 |
| MERCK & CO INC | 16 | 1997–2003 |
| JAPAN TOBACCO INC | 4 | 2005–2010 |
| TULARIK INC | 2 | 2004–2005 |
| AFASCI INC | 1 | 2020 |
Locations
| Location | Patents | Span |
|---|---|---|
| San Francisco, California, US | 29 | 2001–2021 |
| Hoboken, New Jersey, US | 14 | 1997–2003 |