Disclosed herein is a solid oral formulation comprising a therapeutically effective amount of a compound of Formula (A) formulated for release of the compound in the intestine, wherein the compound of Formula (A) has the structure: [structure]

Claims

13 · 1 independent · depth 7

13 granted claims

›1.independentA solid oral formulation comprising a therapeutically effective amount of a compound of Formula (A) formulated for release of the compound in the inte…+12

›2.↳ 1The solid oral formulation of claim 1, wherein R2 and R3 are each H.d2+5

›8.↳ 1The solid oral formulation of claim 1, wherein the compound of Formula (A) or a pharmaceutically acceptable solvate, hydrate, or salt thereof is relea…d2

›9.↳ 1The solid oral formulation of claim 1, further comprising at least one coating chosen from enteric coatings and non-enteric differential release coati…d2+1

›11.↳ 1The solid oral formulation of claim 1, wherein the compound of Formula (A) or a pharmaceutically acceptable solvate, hydrate, or salt thereof is relea…d2

›12.↳ 1The solid oral formulation of claim 1, further comprising at least one pharmaceutically acceptable excipient.d2

›13.↳ 1The solid oral formulation of claim 1, wherein the formulation is in the form of a tablet or capsule.d2

Classifications

6 codes

IPC · International Patent Classification

Section A — Human necessities

A61K31/519
A61K9/48
A01N43/90
A61K45/06
A61K31/00

Section C — Chemistry; metallurgy

C07D487/04

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File wrapper

Pendency

1.7 y

636 days filing → grant

Office actions

after a restriction

Responses

no RCE

Interviews

examiner interview summaries

Examiner

Jeffrey H Murray

art unit 1624 · TC 1600

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Citations: 444 back · 0 forward

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Priority chain

2 priority documents

Priority

22 Sep 2006

earliest claimed

›Priority documents — 2

Type	Document	Date
provisional	US 60826720	22 Sep 2006
related publication	US 20140212485 A1	31 Jul 2014

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