›1.independentA compound of formula I ##STR41## in which R.sup.1 is benzoyl or t-butyloxycarbonyl; R.sup.2 is acetoxy, hydrogen or hydroxy; and the wavy line indica…+12
A compound of formula I ##STR41## in which R.sup.1 is benzoyl or t-butyloxycarbonyl; R.sup.2 is acetoxy, hydrogen or hydroxy; and the wavy line indicates either the .alpha.- or the .beta.-configuration.
›2.↳ 1A compound of claim 1 that is 7-fluorotaxol.d2+2
A compound of claim 1 that is 7-fluorotaxol.
›3.↳ 2The compound of claim 2 that is 7.alpha.-fluorotaxol.d3
The compound of claim 2 that is 7.alpha.-fluorotaxol.
›4.↳ 2The compound of claim 2 that is 7.beta.-fluorotaxol.d3
The compound of claim 2 that is 7.beta.-fluorotaxol.
›5.↳ 1A compound of claim 1 that is N-debenzoyl-N-t-butoxycarbonyl-7-fluorotaxol.d2+2
A compound of claim 1 that is N-debenzoyl-N-t-butoxycarbonyl-7-fluorotaxol.
›6.↳ 5The compound of claim 5 that is N-debenzoyl-N-t-butoxycarbonyl-7.alpha.-fluorotaxol.d3
The compound of claim 5 that is N-debenzoyl-N-t-butoxycarbonyl-7.alpha.-fluorotaxol.
›7.↳ 5The compound of claim 5 that is N-debenzoyl-N-t-butoxycarbonyl-7.beta.-fluorotaxol.d3
The compound of claim 5 that is N-debenzoyl-N-t-butoxycarbonyl-7.beta.-fluorotaxol.
›8.↳ 1A compound of claim 1 that is 7-fluoro-10-desoxytaxol.d2+2
A compound of claim 1 that is 7-fluoro-10-desoxytaxol.
›9.↳ 8The compound of claim 8 that is 7-fluoro-10-desoxytaxol.d3
The compound of claim 8 that is 7-fluoro-10-desoxytaxol.
›10.↳ 8The compound of claim 8 that is 7.beta.-fluoro-10-desoxytaxol.d3
The compound of claim 8 that is 7.beta.-fluoro-10-desoxytaxol.
›11.↳ 1A compound of claim 1 that is 7-fluoro-10-desacetyltaxol.d2+2
A compound of claim 1 that is 7-fluoro-10-desacetyltaxol.
›12.↳ 11The compound of claim 11 that is 7.alpha.-fluoro-10-desacetyltaxol.d3
The compound of claim 11 that is 7.alpha.-fluoro-10-desacetyltaxol.
›13.↳ 11The compound of claim 11 that is 7.beta.-fluoro-10-desacetyltaxol.d3
The compound of claim 11 that is 7.beta.-fluoro-10-desacetyltaxol.
›14.independentmultiple · 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13A pharmaceutical formulation which comprises as an active ingredient a compound as claimed in any one of claims 1 to 13 associated with one or more ph…
Multiple dependency — claims 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13. Shown here under ; it stands on every one of them.
A pharmaceutical formulation which comprises as an active ingredient a compound as claimed in any one of claims 1 to 13 associated with one or more pharmaceutically acceptable carriers, excipients or diluents therefor.
›15.independentmultiple · 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13A method for treating mammalian tumors which comprises administering to a mammal a tumor sensitive amount of a compound as claimed in any one of claim…
Multiple dependency — claims 1, 2, 3, 4, 5, 6, 7, 8, 9, 10, 11, 12, 13. Shown here under ; it stands on every one of them.
A method for treating mammalian tumors which comprises administering to a mammal a tumor sensitive amount of a compound as claimed in any one of claims 1 to 13.
›16.independentA fluoro baccatin III of formula IV ##STR42## in which the wavy line indicates either the .alpha.- or the .beta.-configuration.+2
A fluoro baccatin III of formula IV ##STR42## in which the wavy line indicates either the .alpha.- or the .beta.-configuration.
›17.↳ 16The fluoro baccatin III of claim 16 in which fluorine is in the .alpha.-configuration.d2
The fluoro baccatin III of claim 16 in which fluorine is in the .alpha.-configuration.
›18.↳ 16The fluoro baccatin III of claim 16 in which fluorine is in the .beta.-configuration.d2
The fluoro baccatin III of claim 16 in which fluorine is in the .beta.-configuration.
